ETC-1002

Catalog No.: A15815

ACL inhibitor and AMPK activator

ETC-1002

ETC-1002 Chemical Structure

CAS NO. 738606-46-7

ETC-1002 is a novel, first-in-class, orally available, once-daily LDL-C lowering small molecule; activator of hepatic AMP-activated protein kinase (AMPK); also has potent inhibitory activity against hepatic ATP-citrate lyase(IC50=29 uM).

Availability: In stock

Package Price Qty
5 mg
$55.00
10 mg
$80.00
25 mg
$180.00
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Biological Activity

ETC-1002 is a novel, first-in-class, orally available, once-daily LDL-C lowering small molecule; activator of hepatic AMP-activated protein kinase (AMPK); also has potent inhibitory activity against hepatic ATP-citrate lyase(IC50=29 uM).
Targets
AMPK
In vitro DMSO 61 mg/mL (177.07 mM)
Water Insoluble
Ethanol Insoluble
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 29.03 mL 145.14 mL 290.28 mL
0.5 mM 5.81 mL 29.03 mL 58.06 mL
1 mM 2.9 mL 14.51 mL 29.03 mL
5 mM 0.58 mL 2.9 mL 5.81 mL

*The above data is based on the productmolecular weight 344.49. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15815
Actions Inhibitor, Activator
CAS No. 738606-46-7
Formula C19H36O5
M. Wt 344.49
Purity >98%
Synonyms ESP-55016, ETC1002, ETC 1002
SMILES CC(C)(CCCCCC(CCCCCC(C)(C)C(=O)O)O)C(=O)O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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