Fimasartan

Catalog No.: A17477

non-peptide angiotensin II receptor antagonist

Fimasartan

Fimasartan Chemical Structure

CAS NO. 247257-48-3

Fimasartan is a non-peptide angiotensin II receptor antagonist (ARB) used for the treatment of hypertension and heart failure. Through oral administration, fimasartan blocks angiotensin II receptor type 1 (AT1 receptors), reducing pro-hypertensive actions of angiotensin II, such as systemic vasoconstriction and water retention by the kidneys.

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5 mg

Regular Price: $50.00

Special Price $40.00

10 mg

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50 mg

Regular Price: $150.00

Special Price $120.00

100 mg

Regular Price: $240.00

Special Price $192.00

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Biological Activity

Fimasartan is a non-peptide angiotensin II receptor antagonist (ARB) used for the treatment of hypertension and heart failure. Through oral administration, fimasartan blocks angiotensin II receptor type 1 (AT1 receptors), reducing pro-hypertensive actions of angiotensin II, such as systemic vasoconstriction and water retention by the kidneys.
In vitro DMSO 97 mg/mL (193.36 mM)
Ethanol 23 mg/mL (45.85 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 19.93 mL 99.67 mL 199.34 mL
0.5 mM 3.99 mL 19.93 mL 39.87 mL
1 mM 1.99 mL 9.97 mL 19.93 mL
5 mM 0.4 mL 1.99 mL 3.99 mL

*The above data is based on the productmolecular weight 501.65. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A17477
Actions Antagonist
CAS No. 247257-48-3
Formula C27H31N7OS
M. Wt 501.65
Purity >98%
Synonyms BR-A657; BR A657; BRA657; BRA 657; Fimasartan. brand name: Kanarb.
SMILES S=C(N(C)C)CC1=C(C)N=C(CCCC)N(CC2=CC=C(C3=CC=CC=C3C4=NN=NN4)C=C2)C1=O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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