Fig. 1 · Structure
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LEI-101 free base
Cat. No.
A73392
CAS
1228660-00-1
Endogenous Metabolite
LEI-101 free base is a selective and orally bioavailable agonist of the CB2 receptor, primarily targeting inflammation and oxidative stress-related conditions. It demonstrates a binding potency to CB2 receptors that is approximately 100 times greater than its affinity for CB1 receptors, with a pEC50 value of 8. The compound’s pharmacological profile suggests potential applications in the treatment of diseases such as kidney disease, making it valuable in therapeutic research.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Agonist |
| CAS Number | 1228660-00-1 |
| Applications | Endogenous Metabolite |
| Formula | C23H25FN4O4S |
| Molecular Weight | 472.53 |
| SMILES | O=C1N(C(CN1CC2=CC=C(C=C2)C3=NC(CN(CC4)CCS4(=O)=O)=C(C=C3)F)=O)C5CC5 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.