Lestaurtinib

Catalog No.: A11274

multi-kinase inhibitor

Lestaurtinib

Lestaurtinib Chemical Structure

CAS NO. 111358-88-4

Lestaurtinib (CEP-701;KT-5555) is a multi-kinase inhibitor with potent activity against the Trk family of receptor tyrosine kinases. Lestaurtinib inhibits JAK2, FLT3 and TrkA with IC50s of 0.9, 3 and less than 25 nM, respectively.

Availability: In stock

Package Price Qty
5 mg
$405.00
10 mg
$698.00
50 mg
$2,070.00
100 mg
$4,140.00
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Biological Activity

Lestaurtinib (CEP-701;KT-5555) is a multi-kinase inhibitor with potent activity against the Trk family of receptor tyrosine kinases. Lestaurtinib inhibits JAK2, FLT3 and TrkA with IC50s of 0.9, 3 and less than 25 nM, respectively.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.76 mL 113.78 mL 227.55 mL
0.5 mM 4.55 mL 22.76 mL 45.51 mL
1 mM 2.28 mL 11.38 mL 22.76 mL
5 mM 0.46 mL 2.28 mL 4.55 mL

*The above data is based on the productmolecular weight 439.46. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11274
Actions Inhibitor
M. Wt 439.46
Formula C26H21N3O4
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 111358-88-4
Synonyms CEP-701, CEP701, CEP701; KT-5555, KT5555, KT 5555
SMILES O=C(NC1)C2=C1C3=C(C4=C52)N(C6=C3C=CC=C6)[[email protected]@]([[email protected]@](O)(CO)C7)(C)O[[email protected]]7N4C8=C5C=CC=C8

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