MG149

Catalog No.: A14267

KAT5 (Tip60) HAT inhibitor

MG149

MG149 Chemical Structure

CAS NO. 1243583-85-8

MG149 is a potent histone acetyltransferase inhibitor with IC50 of 74 uM and 47 uM for Tip60 and MOF.

Availability: In stock

Package Price Qty
5 mg
$100.00
10 mg
$180.00
25 mg
$334.00
10mM * 1mL in DMSO
$127.00
Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

MG149 is a potent histone acetyltransferase inhibitor with IC50 of 74 uM and 47 uM for Tip60 and MOF.
Targets
MOF Tip60
47 μM74 μM
In vitro DMSO 63 mg/mL (185.03 mM)
Water 63 mg/mL (185.03 mM)
Ethanol Insoluble
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 29.37 mL 146.86 mL 293.72 mL
0.5 mM 5.87 mL 29.37 mL 58.74 mL
1 mM 2.94 mL 14.69 mL 29.37 mL
5 mM 0.59 mL 2.94 mL 5.87 mL

*The above data is based on the productmolecular weight 340.46. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A14267
Actions Inhibitor
CAS No. 1243583-85-8
Formula C22H28O3
M. Wt 340.46
Solubility DMSO
Purity >98%
Synonyms MG 149,MG-149
SMILES CCCCCCCC1=CC=C(C=C1)CCC2=C(C(=CC=C2)O)C(=O)O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Product Tags

Product Tags

Other people marked this product with these tags:

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy MG149 | MG149 Supplier | purchase | cost | manufacturer | order | distributor | buy 1243583-85-8| 1243583-85-8 Supplier | purchase 1243583-85-8 | 1243583-85-8 cost | 1243583-85-8 manufacturer | order 1243583-85-8 | 1243583-85-8 distributor
Rewards