Name: GABAA Modulator I
Brand: Adooq Bioscience
SKU: A22646
Rating: 5 (288 reviews)

Catalog No.

Product Name

Application

Product Information

Citations

A13449

Lorediplon

GABAA receptor modulator

Lorediplon is a novel non-benzodiazepine, hypnotic drug acting as a GABAA receptor modulator,

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A13769

Indiplon

GABAA receptor modulator

Indiplon is a pyrazolopyrimidine that acts as a high-affinity positive allosteric modulator of the GABAA receptor, potentiating GABA-activated chloride currents in a dose-dependent and reversible manner.

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A15939

CTP354

GABA(A) modulator

CTP354 a novel deuterated subtype-selective GABA(A) modulator.

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A19292

NEO 376

5-HT1 receptor modulator

NEO 376 is a selective modulator of 5-HT1 receptor, GABA receptor and dopamine receptor, with anti-psychotic actively.

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A19295

Loreclezole

GABAA receptor modulator

Loreclezole, an antiepileptic compound, is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit containing receptors.

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A19337

ONO-8590580

GABAA α5 modulator

ONO-8590580 is a GABAA α5 negative allosteric modulator.

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A19357

LAU159

α1β3 GABA(A) receptor modulator

LAU159 is a functionally selective positive modulator of α1β3 GABA(A) receptor with an EC50 of 2.2 μM.

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A20684

AZD-6280

GABAA(α2/3) receptor modulator

AZD-6280 is a selective GABAA(α2/3) receptor modulator, used for treatment of generalized anxiety disorder.

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A21321

Basmisanil

GABAAα5 modulator

Basmisanil is a highly selective GABAAα5 negative allosteric modulator.

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A21425

NS11394

GABA(A) receptor modulator

NS11394 is a potent and subtype-selective GABA(A) receptor-positive modulator; possesses a functional efficacy selectivity profile of alpha(5) > alpha(3) > alpha(2) > alpha(1) at GABA(A) alpha subunit-containing receptors.

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A22188

SSD114 hydrochloride

GABAB receptor positive allosteric modulator

SSD114 hydrochloride is a novel GABAB receptor positive allosteric modulator.

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A22247

Imidazenil

GABA-A modulator

Imidazenil is a GABA-A modulator that blocks the sedative effects without lowering the convulsion threshold.

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A22632

SJM-3

positive allosteric modulator of different isoforms of the GABAA receptor

SJM-3 is a positive allosteric modulator of different isoforms of the GABAA receptor. SJM-3 binds at the high-affinity benzodiazepine binding site at the α+/γ- subunit interface.

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A22646

GABAA Modulator I

modulator of the GABAA receptor complex

GABAA Modulator I is novel modulator of the GABAA receptor complex, and in particular for combating anxiety and related diseases.

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GABA Receptors