PD 123319 ditrifluoroacetate

Catalog No.: A13201

angiotensin AT2 receptor antagonist

PD 123319 ditrifluoroacetate

PD 123319 ditrifluoroacetate Chemical Structure

CAS NO. 130663-39-7

PD 123319 ditrifluoroacetate is a potent, selective, non-peptide angiotensin AT2 receptor antagonist. IC50 values are 34 and 210 nM in rat adrenal tissue and brain respectively.

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10 mg
$120.00
25 mg
$240.00
50 mg
$400.00
100 mg
$700.00
10mM * 1mL in DMSO
$140.00
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  • Dao-Lai Zhang, .et al. Gq activity- and β-arrestin-1 scaffolding-mediated ADGRG2/CFTR coupling are required for male fertility, eLife, 2018, 7: e33432 PMID: 29393851

Biological Activity

PD 123319 ditrifluoroacetate is a potent, selective, non-peptide angiotensin AT2 receptor antagonist. IC50 values are 34 and 210 nM in rat adrenal tissue and brain respectively.
Targets
AT2 receptor
34 nM
In vitro (25°C) DMSO 100 mg/mL (196.61 mM)
Water 100 mg/mL (196.61 mM)
Ethanol 100 mg/mL (196.61 mM)
In vivo Saline 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 13.57 mL 67.87 mL 135.75 mL
0.5 mM 2.71 mL 13.57 mL 27.15 mL
1 mM 1.36 mL 6.79 mL 13.57 mL
5 mM 0.27 mL 1.36 mL 2.71 mL

*The above data is based on the productmolecular weight 736.67. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A13201
Actions Antagonist
M. Wt 736.67
Formula C31H32N4O3.2CF3CO2H
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 130663-39-7
Synonyms PD123319, PD-123319
SMILES CC1=C(C=CC(=C1)CN2C=NC3=C2C[[email protected]](N(C3)C(=O)C(C4=CC=CC=C4)C5=CC=CC=C5)C(=O)O)N(C)C

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