TCS PIM-1 1

Catalog No.: A15369

Pim-1 Kinase Inhibitor

TCS PIM-1 1

TCS PIM-1 1 Chemical Structure

CAS NO. 491871-58-0

TCS PIM-1 1 is a potent and selective ATP-competitive Pim-1 kianse inhibitor with IC50 of 50 nM, displays good selectivity over Pim-2 and MEK1/MEK2(IC50s >20,000 nM).

Availability: In stock

Package Price Qty
10 mg
$110.00
50 mg
$270.00
100 mg
$500.00
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Biological Activity

TCS PIM-1 1 is a potent and selective ATP-competitive Pim-1 kianse inhibitor with IC50 of 50 nM, displays good selectivity over Pim-2 and MEK1/MEK2(IC50s >20,000 nM).
In vitro DMSO 70 mg/mL (190.63 mM)
Water <1 mg/mL
Ethanol <1 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 27.23 mL 136.17 mL 272.33 mL
0.5 mM 5.45 mL 27.23 mL 54.47 mL
1 mM 2.72 mL 13.62 mL 27.23 mL
5 mM 0.54 mL 2.72 mL 5.45 mL

*The above data is based on the productmolecular weight 367.2. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15369
Actions Inhibitor
CAS No. 491871-58-0
Formula C18H11BrN2O2
M. Wt 367.2
Solubility DMSO
Purity >98%
Synonyms SC 204330, TCS PIM 1-1
SMILES C1=CC=C(C=C1)C2=C(C(=O)NC(=C2)C3=C(C=CC(=C3)Br)O)C#N
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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