VP3.15 dihydrobromide

Catalog No.: A21789

PDE7/GSK3 inhibitor

VP3.15 dihydrobromide

VP3.15 dihydrobromide Chemical Structure

CAS NO. 1281681-33-1

VP3.15 dihydrobromide is a potent, orally bioavailable and CNS-penetrant dual phosphodiesterase (PDE)7- glycogen synthase kinase (GSK)3 inhibitor, with IC50s of 1.59 μM and 0.88 μM for PDE7 and GSK-3, respectively.

Availability: In stock

Package Price Qty
5 mg
$135.00
10 mg
$233.00
50 mg
$690.00
100 mg
$1,380.00
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Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

VP3.15 dihydrobromide is a potent, orally bioavailable and CNS-penetrant dual phosphodiesterase (PDE)7- glycogen synthase kinase (GSK)3 inhibitor, with IC50s of 1.59 μM and 0.88 μM for PDE7 and GSK-3, respectively.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 18.93 mL 94.64 mL 189.29 mL
0.5 mM 3.79 mL 18.93 mL 37.86 mL
1 mM 1.89 mL 9.46 mL 18.93 mL
5 mM 0.38 mL 1.89 mL 3.79 mL

*The above data is based on the productmolecular weight 528.3. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21789
Actions Inhibitor
CAS No. 1281681-33-1
Formula C20H24Br2N4OS
M. Wt 528.3
Purity >98%
SMILES [H]Br.[H]Br.N1(CC/N=C2N=C(C3=CC=CC=C3)N(C4=CC=CC=C4)S/2)CCOCC1
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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