Amino acid transporter

BCH is an inhibitor of L-type amino acid transporter LAT1. Suppresses growth and induces apoptosis via activation of caspases in KB, Saos2 and C6 cancer cell lines.

RG1678 (Bitopertin) is a potent and noncompetitive glycine reuptake inhibitor (GlyT1).

RG1678 (Bitopertin) is a potent and noncompetitive glycine reuptake inhibitor (GlyT1).

Amoxapine is a tricyclic dibenzoxazepine (an N-aryl piperazine) which acts similarly to several other tricyclic antidepressants, amoxapine inhibits GLYT2a transport activity with IC50 of 92 μM.

Sarcosine is a glycine transporter type 1 (GlyT) inhibitor and an N-methyl-D-aspartate (NMDA) receptor co-agonist at the glycine binding site.

V-9302 is a competitive antagonist of transmembrane glutamine flux.

JPH203 is a potent and selective L-type amino acid transporter 1 (LAT-1) inhibitor.

GPNA hydrochloride is a well known substrate of the enzyme γ-glutamyltransferase (GGT). GPNA hydrochloride is a specific glutamine (Gln) transporter ASCT2 inhibitor.

Sarcosine ethyl ester hydrochloride is a Glycine derivative.