Tubastatin A HCl

Catalog No.: A11042

HDAC6 inhibitor

Tubastatin A HCl Chemical Structure

CAS NO. 1310693-92-5, 1239262-52-2

Tubastatin A is a potent and selective HDAC6 inhibitor with IC50 of 15 nM in a cell-free assay. It is selective against all the other isozymes (1000-fold) except HDAC8 (57-fold).

Availability: In stock

Package Price Qty
10 mg
$60.00
25 mg
$80.00
50 mg
$90.00
100 mg
$150.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

Tubastatin A is a potent and selective HDAC6 inhibitor with IC50 of 15 nM in a cell-free assay. It is selective against all the other isozymes (1000-fold) except HDAC8 (57-fold).
Targets
Target Value
HDAC6IC50: 15nM
HDAC8IC50: 854nM
HDAC1IC50: 16.4μM
HDAC2IC50: >30μM
HDAC3IC50: >30μM
HDAC4IC50: >30μM
HDAC5IC50: >30μM
HDAC7IC50: >30μM
HDAC9IC50: >30μM
HDAC10IC50: >30μM
HDAC11IC50: >30μM
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 26.89 mL 134.44 mL 268.89 mL
0.5 mM 5.38 mL 26.89 mL 53.78 mL
1 mM 2.69 mL 13.44 mL 26.89 mL
5 mM 0.54 mL 2.69 mL 5.38 mL

*The above data is based on the productmolecular weight 371.9 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11042
Actions Inhibitor
M. Wt 371.9
Formula C20H21N3O2.HCl
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1310693-92-5, 1239262-52-2
Synonyms N/A
SMILES CN1CCC2=C(C1)C3=CC=CC=C3N2CC4=CC=C(C=C4)C(=O)NO.Cl

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