GABA Receptors



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Catalog No. Product Name Application Product Information
A12590

(+)-Bicuculline

GABAA antagonist
(+)-Bicuculline is a classical GABAA antagonist.
A13696

2-Hydroxysaclofen

GABAB receptors antagonist
2-Hydroxysaclofen is a potent and selective antagonist at GABAB receptors.
A13726

AWD 131-138

GABAA receptor agonist
AWD 131-138 is a new low-affinity partial benzodiazepine receptor agonist with potent anticonvulsant and anxiolytic properties in rodent models.
A10121 SALE

Baicalin

HIV-1 production Inhibitor
Baicalin is a known prolyl endopeptidase inhibitor and affects the GABA receptors.
A15939

CTP354

GABA(A) modulator
CTP354 a novel deuterated subtype-selective GABA(A) modulator.
A10397 SALE

Flumazenil

Benzodiazepine antagonist
Flumazenil, an imidazobenzodiazepine derivative, antagonizes the actions of benzodiazepines on the central nervous system. Flumazenil competitively inhibits the activity at the benzodiazepine recognition site on the GABA/benzodiazepine receptor complex. Flumazenil is a weak partial agonist in some animal models of activity, but has little or no agonist activity in humans.
A10412 SALE

Furosemide

-
Furosemide is a non-competitive antagonist at GABAA receptors with ~ 100-fold greater selectivity for α6-containing receptors than α1-containing receptors.
A10413 SALE

Gabapentin

-
Gabapentin (Neurontin) is a pharmaceutical agent, specifically a GABA analogue.
A14004

Picrotoxin

GABAA receptor antagonist
Picrotoxin is a GABAA receptor antagonist. This compound has been shown to increase noradrenaline levels and turnover in the hypothalamus.
A10754

Primidone (Mysoline)

-
Primidone is an anticonvulsant. Potentiates GABAA receptor function.
A10849

SKF 89976A HCl

GABA uptake inhibitor
SKF 89976A hydrochloride is a potent inhibitor of GABA uptake with IC50 of 0.13, 550, 944 and 7210 μM for hGAT-1, rGAT-2, hGAT-3 and hBGT-1 respectively.
A13198

Tiagabine

GABA reuptake inhibitor
Tiagabine is a selective gamma-aminobutyric acid (GABA) reuptake inhibitor.
A15277

Vigabatrin

GABA-transaminase inhibitor
Vigabatrin is a structural analog of the inhibitory neurotransmitter ??-aminobutyric acid (GABA) that irreversibly inhibits the catabolism of GABA by GABA transaminase.
A15441

Vigabatrin

GABA-T inhibitor
Vigabatrin is an antiepileptic drug that inhibits the breakdown of gamma-aminobutyric acid (GABA) by acting as a suicide inhibitor of GABA transaminase (GABA-T).
A12993

Zaleplon

-
Zaleplon is a non-benzodiazepine agent that acts as an agonist at the benzodiazepine site.

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