Flumazenil

Catalog No.: A10397
Benzodiazepine antagonist
Flumazenil, an imidazobenzodiazepine derivative, antagonizes the actions of benzodiazepines on the central nervous system. Flumazenil competitively inhibits the activity at the benzodiazepine recognition site on the GABA/benzodiazepine receptor complex. Flumazenil is a weak partial agonist in some animal models of activity, but has little or no agonist activity in humans.
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Flumazenil 50mg
Special Price $72.00 Regular Price $90.00
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Flumazenil 100mg
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Flumazenil 200mg
Special Price $200.00 Regular Price $250.00
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Flumazenil 500mg
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Prop65 Warning  WARNING: Attention California Residents: This product can expose you to chemicals including Flumazenil , which is known to the State of California to cause cancer and birth defects or other reproductive harm. For more information, go to www.P65Warnings.ca.gov

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Biological Activity
Discription Flumazenil, an imidazobenzodiazepine derivative, antagonizes the actions of benzodiazepines on the central nervous system. Flumazenil competitively inhibits the activity at the benzodiazepine recognition site on the GABA/benzodiazepine receptor complex. Flumazenil is a weak partial agonist in some animal models of activity, but has little or no agonist activity in humans.
Targets
Target Value
Product Information
Catalog Num A10397
Formula C15H14FN3O3
Molecular Weight 303.3
CAS Number 78755-81-4
SMILES CCOC(=O)c1ncn2c1CN(C)C(=O)c1c2ccc(c1)F
Synonyms Ro 15-1788
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility
In vitro DMSO 4 mg/mL (13.18 mM)
Water Insoluble
Ethanol Insoluble
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Preparing Stock Solutions
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 32.97 mL 164.85 mL 329.71 mL
0.5 mM 6.59 mL 32.97 mL 65.94 mL
1 mM 3.3 mL 16.49 mL 32.97 mL
5 mM 0.66 mL 3.3 mL 6.59 mL
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

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