Other inhibitors

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  1. GAGs biosynthesis

    Pro-xylane (Hydroxypropyl tetrahydropyrantriol) is a biologically active C-glycoside in aqueous media, acts as an activator of glycosaminoglycans (GAGs) biosynthesis.
  2. KLC2-SKIP Interaction inhibitor

    Kinesore is an inhibitor of the KLC2-SKIP Interaction.
  3. oral antidiabetic agent

    BM-131246 is an oral antidiabetic agent.
  4. Bencianol is a the semisynthetic flavinoid, with anti-spasmogenic activities.
  5. ST inhibitor

    Lith-O-Asp is a sialytransferase (ST) inhibitor, with IC50s of 12-37 μM.
  6. BRAG2 inhibitor

    Bragsin2 is a potent, selective and noncompetitive nucleotide exchange factor BRAG2 inhibitor, with an IC50 of 3 μM.
  7. ArfGEF BRAG2 inhibitor

    Bragsin1 is a potent, selective and noncompetitive inhibitor of the ArfGEF BRAG2, inhibits Arf GTPase activation, with an IC50 of 3 μM.
  8. Oxyfenamate has anti-anxiety actions for use in anxiety neuroses.
  9. spastin inhibitor

    Spastazoline is a potent and selective spastin (a microtubule-severing AAA protein) inhibitor, with an IC50 of 99 nM for Human spastin. Spastazoline shows no effect on ATPase activity of a recombinant human VPS4.
  10. MTHFD1/MTHFD2 inhibitor

    LY 345899 is a methylene tetrahydrofolate dehydrogenase (MTHFD1; DC301) and MTHFD2 inhibitor with IC50 values of 96 nM and 663 nM, respectively and a Ki of 0.018 μM.
  11. Padsevonil is a potent antiepileptic agent.
  12. Arrhythmias-Targeting Compound 1 is used in the research of arrhythmias, extracted from patent WO 2001028992 A2.
  13. IAA antagonist

    PEO-IAA is an indole-3-acetic acid (IAA) antagonist. PEO-IAA is an auxin antagonist that binds to transport inhibitor response 1/auxin signaling F-box proteins (TIR1/AFBs).
  14. hepcidin production inhibitor

    DS28120313 (compound 32) is an orally hepcidin production inhibitor with an IC50 of 0.093 μM.
  15. Tegadifur is a fluorine-containing and anti-metabolic drug.
  16. rat adenylate kinase II inhibitor

    N6-Methyladenosine 5'-monophosphate disodium salt is an activator of glycogen phosphorylase b, with a Ka value of 22 ?M. N6-Methyladenosine 5'-monophosphate disodium salt is a non-competitive rat adenylate kinase II inhibitor.
  17. aminocryptand ligand

    Octaaminocryptand 1 is an aminocryptand ligand.
  18. Benzyl alcohol is an aromatic alcohol; a colorless liquid with a mild pleasant aromatic odor.
  19. Benzyl benzoate is one of the older preparations used to treat scabies. Scabies is a skin infection caused by the mite sarcoptes scabiei.
  20. Bisacodyl (INN) is a stimulant laxative drug that works directly on the colon to produce a bowel movement.
  21. LH-RH, human is a biochem/physiol Actions LHRH Hypothalamic peptide that stimulates release of gonadotrophins from anterior pituitary, thus regulating reproductive functions.
  22. Anisole methoxybenzene is a colorless liquid with a smell reminiscent of anise seed, and in fact many of its derivatives are found in natural and artificial fragrances.
  23. DBU
    DBU is a chemical compound and belongs to the class of amidine compounds.
  24. Triisopropylsilane is a highly selective reducing agent which can be used to prepare anti-1,2-diols.
  25. Bisoctrizole is a broad-spectrum ultraviolet radiation absorber, absorbing UVB as well as UVA rays. Also a hybrid UV absorber, reflecting and scattering UV.
  26. PDX1 inducer

    BRD7552 is an inducer of transcription factor PDX1, which increases insulin expression.
  27. (Z)-2-decenoic acid is an unsaturated short chain fatty acid that is secreted by P. aeruginosa and induces a disp .
  28. 9-Dihydro-13-acetylbaccatin III (9-DHAB III) is an intermediate for taxol analog preparations.
  29. Benfotiamine is a synthetic S-acyl derivative of thiamine (vitamin B1), an antioxidant dietary supplement.
  30. BMX kinase inhibitor

    BMX-IN-1 is a highly selective and potent irreversible inhibitor which target the cysteine residue in the BMX ATP binding domain.
  31. COT/Tpl2 inhibitor

    Cot inhibitor-2 is a COT/Tpl2 inhibitor.
  32. Deferasirox Fe3+ chelate is a rationally-designed oral iron chelator; its main use is to reduce chronic iron overload in patients who are receiving long-term blood transfusions for conditions such as beta-thalassemia and other chronic anemias.
  33. EBE-A22 is a derivative of PD 153035 which can inhibit ErbB-1-phosphorylation, whereas EBE-A22 is inactive.
  34. Etimizol was shown to relieve amnesia effectively in the origin of which there is the hypoxic component (hypobaric hypoxia, actinomycin D, mechanical injury of the brain).
  35. GNG inhibitor

    MB05032 is a special and efficacious GNG inhibitor targeted the AMP binding site of fructose 1,6-bisphosphatase (FBPase) with an IC50 value of 16 nM.
  36. TK inhibitor

    N3PT is a potent and selective transketolase(TK) inhibitor (IC50= 22 nM for Apo-TK) both in vitro and in vivo.
  37. SE inhibitor

    NB-598 is a potent competitive inhibitor of squalene epoxidase (SE). NB-598 suppresses triglyceride biosynthesis through the farnesol pathway.
  38. Pafuramidine is an orally bioavailable prodrug of furamidine, which has clinical activity against Pneumocystis pneumonia.
  39. Pamabron is a common over-the-counter diuretic used for relief of menstrual-associated symptoms.
  40. Retinyl glucoside is a naturally occurring and biologically active metabolites of vitamin A, which are found in fish and mammals.
  41. sodium 4-pentynoate is a alkynylacetate analogue; can be metabolically incorporated onto cellular proteins through biosynthetic mechanisms for profiling of acetylated proteins in diverse cell types.
  42. Sodium formononetin-3'-sulfonate is a water-sol. derivate of formononetin.
  43. R18

    14.3.3 proteins Antagonist

    R18, antagonist of 14.3.3 proteins (KD ??? 80 nM). Competitively inhibits 14.3.3-ligand interactions without requiring phosphorylation.
  44. Immunomodulators

    Plumbagin, exhibits cytotoxicity in rodent models of carcinogenesis and carcinoma; has antifungal, antiviral, and antibacterial action.
  45. Morphine-like substance

    Beta-lipotropin (beta-LPH) was found to contain within its C-terminal sequence the primary structure of these peptides.
  46. Cell adhesion inhibitor

    K-7174 is a novel cell adhesion inhibitor; inhibits the expression of vascular cell adhesion molecule-1 (VCAM-1) induced by either IL-1beta or TNF-alpha.
  47. Cell adhesion inhibitor

    K-7174 dihydrochloride is a novel cell adhesion inhibitor; inhibits the expression of vascular cell adhesion molecule-1 (VCAM-1) induced by either IL-1beta or TNF-alpha.
  48. DNA repair inhibitor

    KRX-0402 is a small molecule that was specifically designed to block the DNA repair protein, MGMT. MGMT confers resistance to certain alkylating agents, such as temozolomide and BCNU, that are commonly used to treat brain cancer, melanoma and non-Hodgkin?€?s lymphoma.
  49. Finafloxacin hydrochloride is a fluoroquinolone compound.

Items 851-900 of 980

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