CaMK

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Catalog No.
Product Name
Application
Product Information
Product Citation
  1. α-adrenergic (AR) antagonist/CaM inhibitor

    Phenoxybenzamine is a cell-permeable, non-specific, irreversible α-adrenergic (AR) antagonist that also acts as an CaM inhibitor.
  2. CaM kinase II inhibitor

    KN-62 is a selective, cell-permeable inhibitor of CaM kinase II.
  3. PKD inhibitor

    CID 2011756 is a protein kinase D (PKD) inhibitor (IC50 values are 0.6, 0.7 and 3.2 μM for PKD2, PKD3 and PKD1 respectively).
  4. PKD inhibitor

    kb NB 142-70 is a selective protein kinase D (PKD) inhibitor (IC50 values are 28.3, 58.7 and 53.2 nM for PKD1, 2 and 3 respectively).
  5. CaM kinase II inhibitor

    KN-93 is an inhibitor of multifunctional Ca++/calmodulin-dependent protein kinase.
  6. eEF2K (CAMKIII) inhibitor

    A-484954 is a potent, selective inhibitor of eukaryotic longation factor-2 kinase (eEF2K).
  7. PKD inhibitor

    CID755673 is a potent PKD inhibitor with IC50s of 182 nM, 280 nM and 227 nM for PKD1, PKD2 and PKD3, respectively.
  8. PKD1 inhibitor

    CID797718 is a structural analog of CID755673 (Adooq Catalog No. A13804). It was a 10-time less potent PKD1 inhibitor with an IC50 value of 7.0 +/-0.8 uM.
  9. CaMK/Phosphorylase inhibitor

    K252a is a highly potent cell permeable inhibitor of CaM kinase and phosphorylase kinase (IC50 = 1.8 and 1.7 nmol/L, respectively).
  10. CaMKII inhibitor

    KN-93 Phosphate is a potent and specific inhibitor of Ca2+/calmodulin-dependent protein kinase II (CaMKII) with Ki of 0.37 μM, no remarkable inhibitory effects on APK, PKC, MLCK or Ca2+-PDE activities.
  11. eEF-2 inhibitor

    NH125 is a selective eEF-2 kinase inhibitor.
  12. CaMK-II Inhibitor

    KN-92 is an inactive derivative of KN-93. KN-93 is a selective inhibitor of Ca2+/calmodulin-dependent kinase II (CaMKII), competitively blocking CaM binding to the kinase (Ki = 370 nM).
  13. CaMK-II Inhibitor

    KN-92 hydrochloride is a negative control for KN-93.
  14. CaMKII inhibitor

    KN-92 is an inactive derivative of KN-93. KN-93 is a selective inhibitor of Ca2+/calmodulin-dependent kinase II (CaMKII), competitively blocking CaM binding to the kinase (Ki = 370 nM).
  15. PKD Inhibitor

    CRT-0066101, potent inhibitor of protein kinase D (PKD); inhibits all PKD isoforms (IC50 values are 1, 2 and 2.5 nM for PKD1, PKD3 and PKD2 respectively).
  16. CaMKK inhibitor

    STO-609 is a cell-permeable inhibitor of calcium/calmodulin-dependent kinase kinases (CaMKK) isoforms CaMKKα and CaMKKβ (Ki = 80 and 15 ng/ml, respectively).
  17. CaMK antagonist

    Calmidazolium chloride (R 24571) is a calmodulin (CaMK) antagonist, antagonizing CaM-dependent phosphodiesterase and calmodulin-induced activation of erythrocyte Ca2+-transporting ATPase with IC50s of 0.15 and 0.35 μM, respectively. Also in anti-cancer research. Calmidazolium binds to CaMK with a Kd of 3 nM.
  18. DCP-LA (FR236924), a linoleic acid derivative, selectively and directly activates PKCε.
  19. calmodulin inhibitor

    Metofenazate is a selective calmodulin inhibitor.
  20. CaMKII inhibitor

    Rimacalib is a Ca2+/calmodulin-dependent protein kinase II (CaMKII) inhibitor, with IC50s of ~1 μM for CaMKIIα to ~30 μM for CaMKIIγ.
  21. CaM-KK inhibitor

    STO-609 is a selective and cell-permeable inhibitor of the Ca2+/calmodulin-dependent protein kinase kinase (CaM-KK), with Ki values of 80 and 15 ng/mL for recombinant CaM-KKα and CaM-KKβ, respectively.
  22. CaMKII inhibitor

    CaMKII-IN-1 is a potent and highly selective CaMKII inhibitor with IC50 of 63 nM.
  23. calmodulin inhibitor

    Zaldaride maleate (CGS-9343B) is a potent and selective inhibitor of calmodulin.
  24. CaMK-II inhibitor

    KN-93 phosphate is a novel membrane-permeant synthetic inhibitor of purified neuronal CaMK-II, with Ki of 370 nM.

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