Target & Activity
| Target | Activity | Value |
|---|---|---|
| PKD1 | IC50 | 28.3 nM |
| PKD3 | IC50 | 53.2 nM |
| PKD2 | IC50 | 58.7 nM |
Cellular Effect
| Cell Line | Activity | Value | Description | Reference |
|---|---|---|---|---|
| LNCaP | IC50 | 2.2 μM | Inhibition of PKD1 autophosphorylation at Ser916 in human PMA-induced LNCAP cells by Western blotting | [PMID: 21617763] |