CRT-0066101

Catalog No.: A16318

PKD Inhibitor

CRT-0066101

CRT-0066101 Chemical Structure

CAS NO. 1883545-60-5

CRT-0066101, potent inhibitor of protein kinase D (PKD); inhibits all PKD isoforms (IC50 values are 1, 2 and 2.5 nM for PKD1, PKD3 and PKD2 respectively).

Availability: In stock

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5 mg

Regular Price: $85.00

Special Price $68.00

10 mg

Regular Price: $155.00

Special Price $124.00

50 mg

Regular Price: $540.00

Special Price $432.00

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Biological Activity

CRT-0066101, potent inhibitor of protein kinase D (PKD); inhibits all PKD isoforms (IC50 values are 1, 2 and 2.5 nM for PKD1, PKD3 and PKD2 respectively).
In vitro DMSO Warmed: 25 mg/mL (60.77 mM)
Water 80 mg/mL (194.49 mM)
Ethanol Warmed: 2 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 24.31 mL 121.56 mL 243.11 mL
0.5 mM 4.86 mL 24.31 mL 48.62 mL
1 mM 2.43 mL 12.16 mL 24.31 mL
5 mM 0.49 mL 2.43 mL 4.86 mL

*The above data is based on the productmolecular weight 411.33. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A16318
Actions Inhibitor
CAS No. 1883545-60-5
Formula C18H22N6O.2HCl
M. Wt 411.33
Purity >98%
Synonyms CRT 0066101, CRT0066101
SMILES Cl.Cl.Cn1cc(cn1)c3cc(c2nc(NC[[email protected]](N)CC)ccn2)c(O)cc3
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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