MAO

Inhibitory Selectivity
Catalog No.Inhibitor Name MAO-AMAO-BMAOOther
A10818Safinamide Mesylate
*
****
A11722Rasagiline Mesylate
***
****
A11885Moclobemide
***
A10690Paeonol
*
**
A13358Tranylcypromine HCl
CYP2A6

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.



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Catalog No. Product Name Application Product Information
A11111 SALE

Rasagiline

MAO B inhibitor
Rasagiline is a selective irreversible inhibitor of MAO-B (monoamine oxidase-B).
A15761 SALE

Olodaterol

MAO inhibitor
Olodaterol is a long acting beta-adrenoceptor agonist used as an inhalation for treating patients with chronic obstructive pulmonary disease (COPD), manufactured by Boehringer-Ingelheim.
A10765 SALE

Quercetin dihydrate (Sophoretin)

MAO-B inhibitor
Quercetin inhibits many enzyme systems including tyrosine protein kinase, phospholipase A2, phosphodiesterases, mitochondrial ATPase, PI 3-kinase and protein kinase C.
A10766 SALE

Quercetin (Sophoretin)

MAO-B inhibitor
Quercetin inhibits many enzyme systems including tyrosine protein kinase, phospholipase A2, phosphodiesterases, mitochondrial ATPase, PI 3-kinase and protein kinase C.
A10454 SALE

Hordenine

MAO-B inhibitor
Hordenine is a phenethylamine alkaloid with antibacterial and antibiotic properties.
A14344

RN-1 2HCl

MAO inhibitor
RN-1 2HCl exhibits selectivity for LSD1 over monoamine oxidase (MAO)-A and MAO-B (IC50 values are 70 nM, 0.51 and 2.79 μM respectively, in a horseradish peroxidase-coupled assay).
A14176

2C-I HCl

MAO inhibitor
Like other 2Cs, 2C-I (hydrochloride) is a monoamine oxidase inhibitor, blocking the breakdown of serotonin and norepinephrine (IC50 values of 79 and 37 uM, respectively), but not dopamine.
A14175

2C-C HCl

MAO inhibitor
2C-C stimulates monoamine receptor activity and inhibits the re-uptake of serotonin and norepinephrine in rat brain synaptosomes (IC50 = 31 and 63 uM, respectively).
A13294

Safinamide

MAO-B inhibitor
Safinamide is a highly selective and reversible monoamine oxidase type B (MAO-B) inhibitor that increases neostriatal dopamine concentration.
A13358 SALE

Tranylcypromine hydrochloride

LSD1/BHC110 & MAO inhibitor
Tranylcypromine hydrochloride is a non-selective MAO-A/B inhibitor.
A13353

Bifemelane HCl

MAO Inhibitor
Bifemelane hydrochloride is an antidepressant MAO inhibitor. Reverses catalepsy induced by tetrabenazine in mice and increases locomotor activity in MPTP-treated marmosets.
A11777

SL251188

MAO-B Inhibitor
SL-251188, an oxazolidinone derivative, was characterized in baboons as a radioligand for the in vivo visualization of MAO-B using positron emission tomography (PET).
A11722

Rasagiline mesylate

Monoamine oxidase inhibitor
Rasagiline is an irreversible inhibitor of monoamine oxidase used as a monotherapy in early Parkinson's disease or as an adjunct therapy in more advanced cases. It is selective for MAO type B over type A by a factor of fourteen.
A10818

Safinamide Mesylate (FCE28073)

MAO Inhibitor
Safinamide Mesylate is mesylate salt of Safinamide, which selectively and reversibly inhibits MAO-B with IC50 of 0.45 μM.
A11885 SALE

Moclobemide

MAO Inhibitor
Moclobemide is a reversible and selective inhibitor of monoamine oxidase A (MAO-A).

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