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5-hydroxymethyl tolterodine (PNU 200577)
Catalog No. A11166 muscarinic receptor antagonist5-hydroxymethyl tolterodine is a metabolite of Tolterodine, a muscarinic receptor antagonist used in the treatment of urinary incontinence.
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BQCA
Catalog No. A17156 BQCA is a highly selective positive allosteric modulator of the M1 muscarinic acetylcholine receptor (mAChR). Learn More -
Metanicotine
Catalog No. A11545 Nicotinic receptor agonistMetanicotine is a neuronal nicotinic receptor agonist, showing high selectivity for the ??4??2 subtype (Ki=26 nM); > 1,000 fold selectivity than ??7 receptors(Ki= 36000 nM). Learn More -
Arecoline
Catalog No. A13071 Arecoline is a cholinergic alkaloid from seeds of the betel nut palm Areca catechu. Learn More -
Oxybutynin
Catalog No. A10684 Oxybutynin(Ditropan) is an anticholinergic medication used to relieve urinary and bladder difficulties. Learn More -
Fesoterodine fumarate (Toviaz)
Catalog No. A10386 AChR antagonistFesoterodine fumarate is a medicine which is used in urinary urgency, reducing the frequency of passing urine and urge urinary incontinence Learn More -
Methscopolamine bromide
Catalog No. A10579 Methscopolamine bromide is a competitive antimuscarinic agent that blocks the binding of acetylcholine at muscarinic acetylcholine receptors (mAChR M). Learn More -
Ipratropium bromide
Catalog No. A10476 Ipratropium bromide is a muscarinic antagonist, bronchodilator, N-Isopropyl salt of atropine. Learn More -
Gallamine triethiodide
Catalog No. A10417 mAChR M2 antagonistGallamine Triethiodide is a mAChR M2 antagonist with pronounced cardioselectivity. Learn More -
Darifenacin
Catalog No. A11987 Darifenacin works by blocking the M3 muscarinic acetylcholine receptor, which is primarily responsible for bladder muscle contractions. Learn More -
Irsogladine
Catalog No. A10480 Rsogladine is an anti-gastric ulcer agent that facilitates gap-junctional intercellular communication through M1 muscarininc acetylcholine receptor binding. Learn More -
Bethanechol chloride
Catalog No. A10180 Muscarinic receptor agonistBethanechol is a parasympathomimetic choline carbamate that selectively stimulates muscarinic receptors without any effect on nicotinic receptors. Learn More -
Orphenadrine citrate
Catalog No. A11712 NMDA receptor antagonistOrphenadrine citrate is a NMDA receptor antagonist with Ki of 6.0 +/- 0.7 μM, HERG potassium channel blocker. Learn More -
SVT-40776 (Tarafenacin)
Catalog No. A10808 muscarinic receptor antagonistSVT-40776 is a novel M3 muscarinic receptor antagonist, for the treatment of overactive bladder. Learn More -
Atropine
Catalog No. A10098 mAChR antagonistAtropine is a competitive antagonist for the muscarinic acetylcholine receptor types M1, M2, M3, M4 and M5. Learn More -
Solifenacin succinate
Catalog No. A11215 muscarinic M3 receptor antagoinstSolifenacin-succinate is a muscarinic M3 receptor antagoinst, used in treatment of urinary incontinence. Learn More -
Tolterodine tartrate (Detrol LA)
Catalog No. A10937 muscarinic receptor antagonistTolterodine tartrate (Detrol LA) is a muscarinic receptor antagonist which is used for the treatment of urinary incontinence. Learn More -
Biperiden HCl
Catalog No. A10147 muscarinic receptor antagonistBiperiden hydrochloride is a muscarinic receptor antagonist that displays some selectivity for the M1 subtype Learn More -
Methoctramine hydrate
Catalog No. A11975 Methoctramine hydrate is a selective M2 muscarinic receptor antagonist at nM concentrations Learn More -
Rocuronium bromide
Catalog No. A10803 AchR antagonistRocuronium Bromide is a competitive AchR antagonist, used in modern anaesthesia. Learn More -
Flavoxate
Catalog No. A12900 muscarinic AChR antagonistFlavoxate binds and inhibits muscarinic receptors, thereby suppressing the micturition reflex and increases urinary bladder capacity by modifying the micturition center in the brain stem. Learn More -
Acetylcholine iodide
Catalog No. A16390 Acetylcholine iodide is a neurotransmitter found at neuromuscular junctions, autonomic ganglia, parasympathetic effector junctions, a subset of sympathetic effector junctions, and at many sites in the central nervous system. Learn More -
Oxotremorine M iodide
Catalog No. A21977 mAChR agonistOxotremorine M iodide is a potent and non-selective muscarinic acetylcholine receptor (mAChR) agonist. Learn More -
Atropine methyl bromide
Catalog No. A18026 mAChR antagonistAtropine methyl bromide, a muscarinic receptor (mAChR) antagonist, is a quaternary ammonium salt of atropine and a mydriatic for dilation of the pupil during ophthalmic examination. It is introduced for relieving pyloric spasm in infants for its highly polar nature. It penetrates less readily into the central nervous system than atropine. Learn More -
Cevimeline hydrochloride
Catalog No. A18092 mAChR agonistCevimeline (Evoxac) Hcl is a parasympathomimetic and muscarinic agonist, with particular effect on M3 receptors; used in the treatment of dry mouth associated with sjogren's syndrome. Learn More -
Anisodamine
Catalog No. A18215 alpha-1 adrenergic receptors / mAChRs inhibitorAnisodamine is an inhibitor of alpha-1 adrenergic receptors and mAChRs isolated from Chinese solanacea plant. Learn More -
Cimetropium Bromide
Catalog No. A18290 mAChR antagonistCimetropium Bromide (DA-3177) is a mAChR antagonist for long-term treatment of irritable bowel syndrome. Learn More -
Darenzepine
Catalog No. A12333 muscarinic receptor inhibitorDarenzepine is a muscarinic receptor inhibitor extracted from patent US 20170095465 A1. Learn More -
Tiotropium Bromide
Catalog No. A10934 muscarinic acetylcholine receptor (mAChR) antagonistTiotropium Bromide (BA679 BR) is a muscarinic acetylcholine receptor (mAChR) antagonist that blocks the binding of the acetylcholine ligand and subsequent opening of the ligand-gated ion channel. Learn More -
Rapacuronium bromide
Catalog No. A21119 mAChR modulatorRapacuronium bromide is an allosteric modulator of muscarinic acetylcholine receptor (mAChR). Learn More -
mAChR-IN-1 hydrochloride
Catalog No. A21398 mAChR antagonistmAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 nM. Learn More -
mAChR-IN-1
Catalog No. A21518 mAChR antagonistmAChR-IN-1 is a potent muscarinic cholinergic receptor(mAChR) antagonist with IC50 of 17 nM. Learn More -
VU0152100
Catalog No. A21769 mAChR M4 potentiatorVU0152100 is a potent and selective allosteric potentiator of M4 mAChR with an EC50 of 380 ?? 93 nM. Learn More -
(Rac)-VU 6008667
Catalog No. A21939 mAChR M5 negative allosteric modulator(Rac)-VU 6008667 is a selective negative allosteric modulator of muscarinic acetylcholine receptor subtype 5 (M5 NAM) (IC50=1.8 μM, pIC50= 5.75), has high CNS penetration. Learn More -
Glycopyrrolate
Catalog No. A12641 muscarinic antagonistGlycopyrrolate is a muscarinic competitive antagonist used as an antispasmodic. Learn More -
Revefenacin
Catalog No. A15986 muscarinic receptor antagonistRevefenacin is potent and selective muscarinic receptor antagonist in development for the treatment of COPD. Learn More -
TBPB
Catalog No. A14205 M1 mAChR agonistTBPB is an allosteric M1 mAChR agonist with EC50 value of 89 nM that regulates amyloid processing and produces antipsychotic-like activity in rats. Learn More -
(-)-Nicotine ditartrate
Catalog No. A13761 (-)-Nicotine ditartrate is a potent agonist of AChR (nicotinic acetylcholine recepto). Learn More -
Imidafenacin
Catalog No. A15490 M3 receptors inhibitorImidafenacin is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM; less potent for M2 receptors(IC50=4.13 nM). Learn More -
Umeclidinium bromide
Catalog No. A15268 Muscarinic receptor antagonistUmeclidinium bromide(GSK573719A) is a muscarinic receptor antagonist which is useful in treatment of chronic obstructive pulmonary disease (COPD). Learn More -
Cevimeline hydrochloride hemihydrate
Catalog No. A15042 M1 agonistCevimeline hydrochloride hemihydrate, a novel muscarinic receptor agonist, is a candidate therapeutic drug for xerostomia in Sjogren's syndrome. Learn More -
PF-3635659
Catalog No. A13548 muscarinic M(3) receptor antagonistPF-3635659 is a potent muscarinic M(3) receptor antagonist. Learn More -
Xanomeline oxalate
Catalog No. A13685 mAChR agonistXanomeline oxalate is a potent agonist of muscarinic acetylcholine receptors (EC50 values are 0.3, 92.5, 5, 52, and 42 nM for M1, M2, M3, M4, and M5, respectively). Learn More -
AF-DX 384
Catalog No. A13856 mAChR antagonistAF-DX 384 is a drug which acts as a selective antagonist of the muscarinic acetylcholine receptors. Learn More -
Nitenpyram
Catalog No. A14229 AchR agonistNitenpyram is a nicotinic acetylcholine receptor (AchR) agonist. Learn More -
Diphenidol HCl
Catalog No. A14244 M2/M3 antagonistDiphenidol HCl is a potent antagonist of muscarinic M2 and M3 receptor with pKb of 6.72 and 7.02. Learn More -
LY2119620
Catalog No. A14217 M2/M4 AChR agonistLY2119620 is a specific, and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors. Learn More -
Catharanthine sulfate
Catalog No. A12161 Catharanthine sulfate is a vinblastine-type alkaloid precursor with antitumor activity. It inhibits AChR by ion channel blocking and desensitization. Learn More -
MK7622
Catalog No. A12835 M1 receptor modulatorMK7622 is a muscarinic M1 receptor positive allosteric modulator. Learn More
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