Pim Kinase



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Catalog No. Product Name Application Product Information
A13203 SALE

AZD1208

pan-Pim kinase inhibitor
AZD1208 is orally available, small molecule inhibitor of PIM kinases with potential antineoplastic activity.
A12896

CX-6258

Pim Inhibitor
CX-6258 is a potent, selective, and orally efficacious pan-Pim kinases inhibitor.
A14275

CX-6258 HCl

Pan-PIM kinase inhibitor
CX-6258 HCl is a potent, orally efficacious pan-Pim kinase inhibitor with IC50 of 5 nM, 25 nM and 16 nM for Pim1, Pim2, and Pim3.
A15055

CX-6258 hydrochloride hydrate

Pim Inhibitor
CX-6258 hydrochloride hydrate is a potent, orally efficacious Pim 1/2/3 kinase(IC50=5 nM/25 nM/16 nM) inhibitor with excellent biochemical potency and kinase selectivity.
A14420

LGB-321 HCl

Pan-PIM kinase inhibitor
LGB-321 HCl is a potent and selective ATP-competitive small molecule inhibitor of PIM kinases (Pan-PIM kinase inhibitor).
A12526 SALE

Losmapimod

Pan-PIM kinase inhibitor
Losmapimod, also know as GW856553 or GW856553X, is a drug developed by GlaxoSmithKline which acts as a selective inhibitor of the enzyme family known as p38 mitogen-activated protein kinases.
A15368

PIM-1 Inhibitor 2

PIM-1 Inhibitor
PIM-1 inhibitor 2 is a potent Pim-1 kinase inhibitor (Ki = 91 nM).
A10838 SALE

SGI-1776 (free base)

PIM Inhibitor
SGI-1776 is a potent and selective inhibitor of Pim kinases that induces apoptosis in CLL and that the mechanism involves Mcl-1 reduction.
A11945 SALE

SMI-4a

Pim Inhibitor
SIM-4a is a Pim kinase inhibitor that blocks mTORC1 activity via activation of AMPK.
A15369 SALE

TCS PIM-1 1

Pim-1 Kinase Inhibitor
TCS PIM-1 1 is a potent and selective ATP-competitive Pim-1 kianse inhibitor with IC50 of 50 nM, displays good selectivity over Pim-2 and MEK1/MEK2(IC50s >20,000 nM).
A11967

TCS PIM-1 4a

Pim inhibitor
TCS PIM-1 4a is a selective and ATP-competitive Pim kinase inhibitor (IC50 values = 24 and 100 nM for Pim-1 and Pim-2, respectively).

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