GDC-0339

Catalog No.: A20920

Pim kinase inhibitor

GDC-0339

GDC-0339 Chemical Structure

CAS NO. 1428569-85-0

GDC-0339 is a potent, orally bioavailable and well tolerated pan-Pim kinase inhibitor, with Kis of 0.03 nM, 0.1 nM and 0.02 nM for Pim1, Pim2 and Pim3, respectively. GDC-0339 is discovered as a potential treatment of multiple myeloma.

Availability: In stock

Package Price Qty
2 mg
$378.00
5 mg
$756.00
10 mg
$1,470.00
50 mg
$4,326.00
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Biological Activity

GDC-0339 is a potent, orally bioavailable and well tolerated pan-Pim kinase inhibitor, with Kis of 0.03 nM, 0.1 nM and 0.02 nM for Pim1, Pim2 and Pim3, respectively. GDC-0339 is discovered as a potential treatment of multiple myeloma.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 21.48 mL 107.41 mL 214.82 mL
0.5 mM 4.3 mL 21.48 mL 42.96 mL
1 mM 2.15 mL 10.74 mL 21.48 mL
5 mM 0.43 mL 2.15 mL 4.3 mL

*The above data is based on the productmolecular weight 465.5. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A20920
Actions Inhibitor
M. Wt 465.5
Formula C20H22F3N7OS
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1428569-85-0
Synonyms GDC0339, GDC 0339
SMILES FC1=CC=CC(F)=C1C2=NC(C(NC3=C(N4CC[[email protected]@H](F)[[email protected]](N)CC4)N(C)N=C3)=O)=C(N)S2

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