AZD-2461

Catalog No.: A12393

PARP Inhibitor

AZD-2461 Chemical Structure

CAS NO. 1174043-16-3

AZD2461 is a novel and potent PARP inhibitor with lower affinity to P-glycoprotein.

Availability: In stock

Package Price Qty
5 mg
$55.00
10 mg
$80.00
25 mg
$150.00
100 mg
$260.00
10mM * 1mL in DMSO
$146.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

AZD2461 is a novel and potent PARP inhibitor with lower affinity to P-glycoprotein.
Targets
PARP
In vitro (25°C) DMSO 79 mg/mL (199.78 mM)
Water <1 mg/mL (<1 mM)
Ethanol 31 mg/mL (78.39 mM)
In vivo 0.5% hydroxyethyl cellulose/0.1% Tween 80 5 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 25.29 mL 126.44 mL 252.89 mL
0.5 mM 5.06 mL 25.29 mL 50.58 mL
1 mM 2.53 mL 12.64 mL 25.29 mL
5 mM 0.51 mL 2.53 mL 5.06 mL

*The above data is based on the productmolecular weight 395.43. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12393
Actions Inhibitor
M. Wt 395.43
Formula C22H22FN3O3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1174043-16-3
Synonyms AZD2461, AZD 2461
SMILES COC1CCN(CC1)C(=O)C2=C(C=CC(=C2)CC3=NNC(=O)C4=CC=CC=C43)F

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