AZD-2461

Catalog No.: A12393

PARP Inhibitor

AZD-2461

AZD-2461 Chemical Structure

CAS NO. 1174043-16-3

AZD2461 is a novel and potent PARP inhibitor with lower affinity to P-glycoprotein.

Availability: In stock

Package Price Qty
5 mg

Regular Price: $55.00

Special Price $44.00

10 mg

Regular Price: $80.00

Special Price $64.00

25 mg

Regular Price: $150.00

Special Price $120.00

100 mg

Regular Price: $260.00

Special Price $208.00

10mM * 1mL in DMSO

Regular Price: $146.00

Special Price $116.80

Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

AZD2461 is a novel and potent PARP inhibitor with lower affinity to P-glycoprotein.
Targets
PARP
In vitro (25°C) DMSO 73 mg/mL (184.61 mM)
Water Insoluble
Ethanol 29 mg/mL (73.33 mM)
In vivo 2% DMSO+40% PEG 300+2% Tween 80+ddH2O 4 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 25.29 mL 126.44 mL 252.89 mL
0.5 mM 5.06 mL 25.29 mL 50.58 mL
1 mM 2.53 mL 12.64 mL 25.29 mL
5 mM 0.51 mL 2.53 mL 5.06 mL

*The above data is based on the productmolecular weight 395.43. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12393
Actions Inhibitor
CAS No. 1174043-16-3
Formula C22H22FN3O3
M. Wt 395.43
Purity >98%
Synonyms AZD2461, AZD 2461
SMILES COC1CCN(CC1)C(=O)C2=C(C=CC(=C2)CC3=NNC(=O)C4=CC=CC=C43)F
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Product Tags

Product Tags

Other people marked this product with these tags:

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy AZD-2461 | AZD-2461 Supplier | purchase | cost | manufacturer | order | distributor | buy 1174043-16-3| 1174043-16-3 Supplier | purchase 1174043-16-3 | 1174043-16-3 cost | 1174043-16-3 manufacturer | order 1174043-16-3 | 1174043-16-3 distributor
Rewards