UPF 1069

Catalog No.: A12750

PARP2 inhibitor

UPF 1069 Chemical Structure

CAS NO. 1048371-03-4

UPF 1069 is a selective poly(ADP-ribose) polymerase (PARP) 2 inhibitor (IC50 values are 0.3 and 8.0 μM for PARP-2 and PARP-1 respectively).

Availability: In stock

Package Price Qty
10 mg
$80.00
25 mg
$150.00
50 mg
$250.00
100 mg
$400.00
10mM * 1mL in DMSO
$81.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

UPF 1069 is a selective poly(ADP-ribose) polymerase (PARP) 2 inhibitor (IC50 values are 0.3 and 8.0 μM for PARP-2 and PARP-1 respectively).
Targets
PARP2 PARP1
0.3 μM8.0 μM
In vitro DMSO 56 mg/mL (200.5 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 35.81 mL 179.03 mL 358.05 mL
0.5 mM 7.16 mL 35.81 mL 71.61 mL
1 mM 3.58 mL 17.9 mL 35.81 mL
5 mM 0.72 mL 3.58 mL 7.16 mL

*The above data is based on the productmolecular weight 279.29. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12750
Actions Inhibitor
M. Wt 279.29
Formula C17H13NO3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1048371-03-4
Synonyms UPF1069, UPF-1069
SMILES C1=CC=C(C=C1)C(=O)COC2=CC=CC3=C2C=CNC3=O

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