AGI-6780

IDH2 R140Q inhibitor

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Catalog No. A12903

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
AGI-6780 5mg A12903-5

Regular Price: $80.00

Special Price: $64.00

AGI-6780 10mg A12903-10

Regular Price: $140.00

Special Price: $112.00

AGI-6780 25mg A12903-25

Regular Price: $280.00

Special Price: $224.00

AGI-6780 50mg A12903-50

Regular Price: $500.00

Special Price: $400.00

AGI-6780 10mM * 1mL in DMSO A12903-10mM-D

Regular Price: $136.00

Special Price: $108.80

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

AGI-6780 is a potent, selective inhibitor of mutant IDH2 with an IC50 value of 23 nM.

AGI-6780

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Chemical Information

Catalog Num A12903
Actions Inhibitor
M. Wt 481.5
Formula C21H18F3N3O3S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1432660-47-3
Synonyms AGI6780
SMILES code C1CC1NS(=O)(=O)C2=CC(=C(C=C2)C3=CSC=C3)NC(=O)NC4=CC=CC(=C4)C(F)(F)F
Chemical Name N-?cyclopropyl-?4-?(3-?thienyl)-?3-?[[[[3-?(trifluoromethyl)phenyl]amino]carbonyl]amino]-?benzenesulfonamide

Biological Activity

Description
AGI-6780 is a potent, selective inhibitor of mutant IDH2 with an IC50 value of 23 nM.
Targets
IDH2 R140Q mutant
23 nM

Solubility

Solubility (25°C)* In vitro DMSO 96 mg/mL (199.37 mM)
Water <1 mg/mL (<1 mM)
Ethanol 96 mg/mL (199.37 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

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