Target & Activity
| Target | Activity | Value |
|---|---|---|
| CDK9/Cyclin T | IC50 | 10 nM |
| CDK5/p35 | IC50 | 13 nM |
| cdk2/cyclin A | IC50 | 47 nM |
| Cdk4/cyclin D1 | IC50 | 100 nM |
| cdk6/cyclin D3 | IC50 | 170 nM |
| Cdk1/cyclin B | IC50 | 210 nM |
| CDK7/Cyclin H/MAT1 | IC50 | 2400 nM |
| GSK3β | IC50 | 89 nM |
8 targets · Scroll to view more