GSK-3787

Catalog No.: A12391
PPAR antagonist
GSK-3787 is a potent and selective peroxisome proliferator-activated receptor δ (PPARδ) antagonist (pIC50 = 6.6).
Grouped product items
Product Name Price Stock Qty
GSK-3787 10mg
$70.00
In stock
GSK-3787 25mg
$140.00
In stock
GSK-3787 50mg
$220.00
In stock
GSK-3787 100mg
$380.00
In stock
GSK-3787 10mM * 1mL in DMSO
$86.00
In stock
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Adooq Products cited in reputable paper
Biological Activity
Discription GSK-3787 is a potent and selective peroxisome proliferator-activated receptor δ (PPARδ) antagonist (pIC50 = 6.6).
Targets
Target Value
Product Information
Catalog Num A12391
Formula C15H12ClF3N2O3S
Molecular Weight 392.78
CAS Number 188591-46-0
SMILES C1=CC(=CC=C1C(=O)NCCS(=O)(=O)C2=NC=C(C=C2)C(F)(F)F)Cl
Synonyms GSK3787, GSK 3787
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility
In vitro DMSO 67 mg/mL (170.58 mM)
Water Insoluble
Ethanol Insoluble
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Preparing Stock Solutions
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 25.46 mL 127.3 mL 254.6 mL
0.5 mM 5.09 mL 25.46 mL 50.92 mL
1 mM 2.55 mL 12.73 mL 25.46 mL
5 mM 0.51 mL 2.55 mL 5.09 mL
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

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