GSK1059615

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mTOR/PI3K Inhibitor

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Catalog No. A10438

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
GSK1059615 5mg A10438-5

Regular Price: $70.00

Special Price: $56.00

GSK1059615 10mg A10438-10

Regular Price: $120.00

Special Price: $96.00

GSK1059615 25mg A10438-25

Regular Price: $250.00

Special Price: $200.00

GSK1059615 50mg A10438-50

Regular Price: $450.00

Special Price: $360.00

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

GSK1059615 is a potent, reversible, ATP-competitive, thiazolidinedione inhibitor of PI3Kα (IC50 = 2 nM).

GSK1059615

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Chemical Information

Catalog Num A10438
Actions Inhibitor
M. Wt 333.4
Formula C18H11N3O2S
Solubility DMSO
Purity >98%
Storage at -20°C 2 years
CAS No. 958852-01-2
Synonyms GSK-1059615
SMILES code C1=CC2=NC=CC(=C2C=C1/C=C\3/C(=O)NC(=O)S3)C4=CC=NC=C4
Chemical Name 5-[[4-(4-Pyridinyl)-6-quinolinyl]methylene]-2,4-thiazolidenedione

Biological Activity

Description
GSK1059615 is a potent, reversible, ATP-competitive, thiazolidinedione inhibitor of PI3Kα (IC50 = 2 nM).
Targets
PI3Kα PI3Kβ PI3Kδ PI3Kγ mTOR
0.4 nM0.6 nM2 nM5 nM12 nM

Solubility

Solubility (25°C)* In vitro DMSO 2 mg/mL (5.99 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

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