Masitinib ( AB1010)

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c-Kit inhibitor

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Catalog No. A10558

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
Masitinib 10mg A10558-10

Regular Price: $50.00

Special Price: $40.00

Masitinib 25mg A10558-25

Regular Price: $90.00

Special Price: $72.00

Masitinib 50mg A10558-50

Regular Price: $110.00

Special Price: $88.00

Masitinib 100mg A10558-100

Regular Price: $168.00

Special Price: $134.40

Masitinib ( AB1010) 10mM * 1mL in DMSO A10558-10mM-D

Regular Price: $50.00

Special Price: $40.00

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

Masitinib (AB1010) is a protein tyrosine kinase inhibitor.

Masitinib ( 	AB1010)

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Chemical Information

Catalog Num A10558
Actions Inhibitor
M. Wt 498.6
Formula C28H30N6OS
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 790299-79-5
Synonyms AB1010, Masivet
SMILES code CC1=C(C=C(C=C1)NC(=O)C2=CC=C(C=C2)CN3CCN(CC3)C)NC4=NC(=CS4)C5=CN=CC=C5
Chemical Name 4-[(4-Methyl-1-piperazinyl)methyl]-N-[4-methyl-3-[[4-(3-pyridinyl)-2-thiazolyl]amino]phenyl]benzamide

Biological Activity

Description
Masitinib (AB1010) is a protein tyrosine kinase inhibitor.
Targets
Target Value
KitIC50: 200nM
LynBIC50: 510nM
PDGFRαIC50: 540nM
PDGFRβIC50: 800nM
Abl1IC50: 1.20μM
c-FmsIC50: 1.48μM
SrcIC50: 1.87μM
HckIC50: 2.0μM
FLT3IC50: >10μM
VEGFR1IC50: >10μM
VEGFR2IC50: >10μM
EGFRIC50: >10μM
FGFR1IC50: >10μM
FGFR3IC50: >10μM
IGF-1RIC50: >10μM
c-MetIC50: >10μM
c-RetIC50: >10μM
JAK2IC50: >10μM
BTKIC50: >10μM
BmxIC50: >10μM
SykIC50: >10μM
FesIC50: >10μM
PKCαIC50: >10μM
Pim1IC50: >10μM
Akt1IC50: >10μM

Solubility

Solubility (25°C) * In vitro DMSO 100 mg/mL (200.54 mM)
Water <1 mg/mL (<1 mM)
Ethanol 4 mg/mL (8.02 mM)
In vivo 1% DMSO/30% polyethylene glycol/1% Tween 80 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

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