Target & Activity
| Target | Activity | Value |
|---|---|---|
| 5-HT2C Receptor | IC50 | 131 nM |
| 5-HT7 Receptor | IC50 | 150 nM |
| 5-HT2A Receptor | IC50 | 478 nM |
| 5-HT2B Receptor | IC50 | 1 μM |
| 5-HT6 Receptor | EC50 | 700 nM |
| 5-HT1A Receptor | EC50 | 3.2 μM |
| D2 Receptor | EC50 | 64 nM |
| D4 Receptor | EC50 | 2 μM |
| D5 Receptor | EC50 | 2.6 μM |
9 targets · Scroll to view more
Cellular Effect
| Cell Line | Activity | Value | Description | Reference |
|---|---|---|---|---|
| B16-4A5 | IC50 | 15.8 μM | Inhibition of melanogenesis in mouse B16-4A5 cells after 72 hrs by spectrophotometry | [PMID: 23270663] |