PIK-93

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PI3K inhibitor

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Catalog No. A10731

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
PIK-93 5mg A10731-5

Regular Price: $70.00

Special Price: $56.00

PIK-93 10mg A10731-10

Regular Price: $120.00

Special Price: $96.00

PIK-93 25mg A10731-25

Regular Price: $220.00

Special Price: $176.00

PIK-93 50mg A10731-50

Regular Price: $380.00

Special Price: $304.00

PIK-93 10mM * 1mL in DMSO A10731-10mM-D

Regular Price: $90.00

Special Price: $72.00

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

PIK 93 selectively inhibits the type III PI 4-kinase enzyme, and small interfering RNA-mediated down-regulation of the individual PI 4-kinase enzymes.

PIK-93

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Chemical Information

Catalog Num A10731
Actions Inhibitor
M. Wt 389.9
Formula C14H16ClN3O4S2
Solubility DMSO
Purity >98%
Storage at -20°C 2 years
CAS No. 593960-11-3
Synonyms PIK93
SMILES code CC1=C(SC(=N1)NC(=O)C)C2=CC(=C(C=C2)Cl)S(=O)(=O)NCCO
Chemical Name N-[5-[4-Chloro-3-[[(2-hydroxyethyl)amino]sulfonyl]phenyl]-4-methyl-2-thiazolyl]acetamide

Biological Activity

Description
PIK 93 selectively inhibits the type III PI 4-kinase enzyme, and small interfering RNA-mediated down-regulation of the individual PI 4-kinase enzymes.
Targets
Target Value
p110γIC50: 16nM
PI4KIIIβIC50: 19nM
p110αIC50: 39nM
DNA-PKIC50: 64nM
p110δIC50: 120nM
C2βIC50: 140nM
hsVps34IC50: 320nM
ATMIC50: 490nM
p110βIC50: 590nM
PI4KIIIαIC50: 1.1μM
mTORC1IC50: 1.38μM
C2αIC50: 16μM
ATRIC50: 17μM
PI4KIIαIC50: >100μM
PI4P5KIαIC50: >100μM
PI4P5KIβIC50: >100μM
PI5P4KIIβIC50: >100μM

Solubility

Solubility (25°C) * In vitro DMSO 78 mg/mL (200.06 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 30% PEG400/0.5% Tween80/5% propylene glycol 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

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