Sitaxsentan sodium (TBC-11251)

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ETA receptor antagonist

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Catalog No. A11564

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
Sitaxsentan sodium (TBC-11251) 5mg A11564-5

Regular Price: $90.00

Special Price: $72.00

Sitaxsentan sodium (TBC-11251) 10mg A11564-10

Regular Price: $160.00

Special Price: $128.00

Sitaxsentan sodium (TBC-11251) 25mg A11564-25

Regular Price: $300.00

Special Price: $240.00

Sitaxsentan sodium (TBC-11251) 50mg A11564-50

Regular Price: $500.00

Special Price: $400.00

Sitaxsentan sodium 10mM * 1mL in DMSO A11564-10mM-D

Regular Price: $145.00

Special Price: $116.00

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

Sitaxentan sodium (TBC-11251) is a selective endothelin receptor-A antagonist with IC50 and Ki of 1.4 nM and 0.43 nM, respectively.

Sitaxsentan sodium (TBC-11251)

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Chemical Information

Catalog Num A11564
Actions Antagonist
M. Wt 476.89
Formula C18H14ClN2NaO6S2
Solubility DMSO
Purity >98%
Storage at -20°C 2 years
CAS No. 210421-74-2
Synonyms N/A
SMILES code CC1=CC2=C(C=C1CC(=O)C3=C(C=CS3)S(=O)(=O)[N-]C4=C(C(=NO4)C)Cl)OCO2.[Na+]
Chemical Name Sodium (4-chloro-3-methyl-1,2-oxazol-5-yl)-[2-[2-(6-methyl-1,3-benzodioxol-5-yl)acetyl]thiophen-3-yl]sulfonylazanide

Biological Activity

Description
Sitaxentan sodium (TBC-11251) is a selective endothelin receptor-A antagonist with IC50 and Ki of 1.4 nM and 0.43 nM, respectively.
Targets
ET-A ET-A
0.43 nM(Ki)1.4 nM

Solubility

Solubility (25°C)* In vitro DMSO 40 mg/mL (83.87 mM)
Water <1 mg/mL (<1 mM)
Ethanol 20 mg/mL (41.93 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

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