Fig. 1 · Structure
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(2R,2R)-PF-07258669
MC4R Antagonist
(2R,2R)-PF-07258669 is an antagonist of the melanocortin 4 receptor (MC4R). It serves as a valuable tool in research aimed at understanding the regulation of appetite and energy expenditure. Its application can aid in elucidating the role of MC4R in metabolic processes and potential therapeutic interventions for obesity and related disorders.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 2755890-68-5 |
| Applications | MC4R Antagonist |
| Formula | C25H27FN6O2 |
| Molecular Weight | 462.52 |
| SMILES | CC(N=C(N1)C(CC[C@@]21CCN(C([C@H](C)C3=C(C=NC(OC)=C3)F)=O)C2)=C4)=C4C5=NC=CC=N5 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.