3-Bromocytisine is a potent agonist of nicotinic acetylcholine receptors (nAChRs), exhibiting IC50 values of 0.28 nM, 0.30 nM, and 31.6 nM for human α4β4, α4β2, and α7 nAChRs, respectively. It demonstrates differential effects on high sensitivity (HS) and low sensitivity (LS) α4β2 nAChRs, with EC50 values of 8 nM and 50 nM, respectively. This compound is valuable for research in neuropharmacology and studies related to nicotine addiction and receptor pharmacodynamics.
3-Bromocytisine is a potent agonist of nicotinic acetylcholine receptors (nAChRs), exhibiting IC50 values of 0.28 nM, 0.30 nM, and 31.6 nM for human α4β4, α4β2, and α7 nAChRs, respectively. It demonstrates differential effects on high sensitivity (HS) and low sensitivity (LS) α4β2 nAChRs, with EC50 values of 8 nM and 50 nM, respectively. This compound is valuable for research in neuropharmacology and studies related to nicotine addiction and receptor pharmacodynamics.
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