Fig. 1 · Structure
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3-Hydroxy darifenacin
M1-5 Muscarinic Receptors Antagonist
3-Hydroxy darifenacin is an antagonist of M1-5 muscarinic receptors, demonstrating Ki values of 17.78, 79.43, 2.24, 36.31, and 6.17 nM in CHO cells. As a metabolite of Darifenacin, it serves as a valuable tool in pharmacological research, particularly in studies focusing on muscarinic receptor signaling and its role in various physiological and pathological processes. Its selective action on muscarinic receptors provides insights into potential therapeutic strategies for disorders influenced by cholinergic signaling.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 206048-82-0 |
| Applications | M1-5 Muscarinic Receptors Antagonist |
| Formula | C28H30N2O3 |
| Molecular Weight | 442.55 |
| SMILES | NC(C(C1=CC=CC=C1)(C2=CC=CC=C2)[C@H]3CN(CC3)CCC4=CC=C(OCC5O)C5=C4)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.