Fig. 1 · Structure
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5-HT2A antagonist 2
5HT2A antagonist
5-HT2A Antagonist 2 is a selective antagonist that targets the 5-HT2A receptor, demonstrating an IC50 value of 14 nM. This compound exhibits favorable chemical stability and retains activity in hepatocyte and plasma environments, while showing negligible cytotoxicity across several cell lines, including VERO, HFL-1, L929, NIH3T3, and CHO-K1. It is suitable for research applications related to neuropharmacology, psychiatric disorders, and other areas involving serotonin receptor modulation.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 2641482-08-6 |
| Applications | 5HT2A antagonist |
| Formula | C30H33ClN4O2 |
| Molecular Weight | 517.06 |
| SMILES | CC1=C(CCN2CC/C(CC2)=C3C(C=CC(Cl)=C4)=C4CCC5=CC=CN=C5\3)C(N(CCCC6O)C6=N1)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.