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5-HT2A inverse agonist-1

5-HT2A Inverse Agonist

5-HT2A inverse agonist-1 is a potent inverse agonist of the 5-HT2A receptor, exhibiting an IC50 of 5.5 nM. This compound demonstrates minimal inhibition of hERG channels, making it a valuable tool in pharmacological research. Its application spans the investigation of neurological diseases, including Parkinson’s disease, facilitating the study of receptor signaling pathways and potential therapeutic interventions.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Inverse Agonist
CAS Number	3028943-38-3
Applications	5-HT2A Inverse Agonist
Formula	C₂₂H₂₅F₅N₄O₂
Molecular Weight	472.45
SMILES	FC(C=C1)=CC=C1CN([C@@H]2[C@@H](CN(CC2)C)F)C(NCC3=CN=C(OCC(F)(F)F)C=C3)=O

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.