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5-HT2CR agonist 2

5-HT2CR Agonist

5-HT2CR Agonist 2 is a selective agonist targeting the 5-HT2C receptor, demonstrating an EC50 of 36 nM. This compound effectively penetrates the blood-brain barrier and exhibits Gq-biased signaling. It has been shown to attenuate MK801-induced hyperlocomotion and reverse hyperlocomotor activity induced by phencyclidine, making it a valuable tool for research into neuropsychiatric disorders and the modulation of dopaminergic activity.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Agonist
CAS Number	2841457-05-2
Applications	5-HT2CR Agonist
Formula	C₁₇H₁₇Cl₂NO₂
Molecular Weight	338.23
SMILES	COC1=C(C=C2C3=C1C4=C(CC3NCC2)C=CC=C4Cl)O.Cl

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.