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5-HT2CR allosteric modulator 1

Positive Ago-allosteric Modulator Of 5HT2CR

5-HT2CR Allosteric Modulator 1 is a selective positive ago-allosteric modulator of the 5-HT2C receptor, exhibiting an EC50 of 8 nM. In addition to its modulating properties, it acts as a selective agonist at the 5-HT2C receptor with an EC50 of 25 nM. This compound has been shown to reduce food intake, making it a valuable tool for research into appetite regulation and related neurobiological pathways.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Modulator
CAS Number	2376501-96-9
Applications	Positive Ago-allosteric Modulator Of 5HT2CR
Formula	C₁₄H₁₄O₃
Molecular Weight	230.26
SMILES	O=C1OC(C2(CCCC2)O)=CC3=C1C=CC=C3

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.