Documents & Downloads

5-HT6/5-HT2AR antagonist-1

5-HT6/5-HT2AR Antagonist

5-HT6/5-HT2AR antagonist-1 is a potent dual antagonist targeting the 5-HT6 and 5-HT2A receptors, exhibiting Ki values of 11 nM and 39 nM, respectively. This compound's inhibition of serotonergic signaling pathways is relevant in the study of neuropsychiatric disorders and cognitive function. Its dual-action mechanism makes it a valuable tool for researchers exploring the therapeutic potential in conditions such as schizophrenia and Alzheimer's disease.

Out of Stock

Free Aliquoting for Your Order

Tell us your preferred amount per vial. We’ll confirm the options.

Specifications

Manufacturer	Adooq Bioscience
Actions	Antagonist
CAS Number	2763654-60-8
Applications	5-HT6/5-HT2AR Antagonist
Formula	C₂₁H₂₆N₆S
Molecular Weight	394.54
SMILES	NC1=NC(N2CCN(C)CC2)=NC(C(C)(SC3=CC=C4C=CC=CC4=C3)C)=N1

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.