Fig. 1 · Structure
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A-794282
mGlu1R Antagonist
A-794282 is a selective antagonist of the metabotropic glutamate receptor 1 (mGlu1R), primarily functioning to modulate pain signaling. This compound exhibits notable analgesic activity, effectively reducing pain behaviors in models of postoperative pain. Caution is advised, as higher doses may produce motor side effects, making it a critical focus for research in pain management and pharmacology.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 869802-44-8 |
| Applications | mGlu1R Antagonist |
| Formula | C19H18N4OS |
| Molecular Weight | 350.44 |
| SMILES | O=C1N(C=NC2=C1SC3=NC=CC(N(C)C)=C23)C4=CC=C(C=C4)CC |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.