Fig. 1 · Structure
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A-850002
mGluR Antagonist
A-850002 is a selective antagonist of metabotropic glutamate receptors (mGluRs) with an IC50 of 27 nM. This compound has been shown to significantly reduce spontaneous pain behavior following skin incision in rodent models. A-850002 is suitable for research applications focused on analgesia and the investigation of pain pathways.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 869802-73-3 |
| Applications | mGluR Antagonist |
| Formula | C18H16N4OS |
| Molecular Weight | 336.41 |
| SMILES | O=C1C2=C(C3=C(C=NC=C3N(C)C)S2)N=CN1C4=CC=C(C)C=C4 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.