Fig. 1 · Structure
Documents & Downloads
α-Casozepine
Anxiolytic
α-Casozepine is an orally bioavailable anxiolytic that targets the benzodiazepine site of the GABAA receptor, exhibiting an IC50 of 88 μM in bovine samples. It demonstrates substantial anxiolytic and anti-stress effects in animals, including cats under unfamiliar conditions and dogs during travel. With proven effectiveness in reducing anxiety responses in rats, α-Casozepine is a valuable tool for research focused on fear, anxiety, and stress-related behaviors.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| CAS Number | 117592-45-7 |
| Applications | Anxiolytic |
| Formula | C60H94N14O16 |
| Molecular Weight | 1267.47 |
| SMILES | [C@H](CC1=CC=C(O)C=C1)(C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@@H](CCCNC(=N)N)C(O)=O)=O)CC(C)C)=O)CC(C)C)=O)CCC(N)=O)=O)CCC(O)=O)=O)CC(C)C)=O)NC(CNC([C@@H](NC([C@H](CC2=CC=C(O)C=C2)N)=O)CC(C)C)=O)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.