Fig. 1 · Structure
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A1AR antagonist 3
A1 Antagonist
A1AR antagonist 3 is a selective antagonist of the adenosine A1 receptor, exhibiting Ki values of 9.69 nM for human A1 and 0.529 nM for rat A1. This compound is valuable for research into neurological diseases, providing insights into the role of A1 receptors in various pathophysiological conditions. Its specificity and potency make it an important tool for studying adenosine signaling and its implications in the central nervous system.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 2413257-73-3 |
| Applications | A1 Antagonist |
| Formula | C25H20N2O3S |
| Molecular Weight | 428.50 |
| SMILES | COC1=CC=C(C=C1)C(NC2=NC(C3=CC=CC=C3)=C(S2)C(C4=CC=C(C=C4)C)=O)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.