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α2C adrenoceptor agonist 1

α2C-adrenoceptor Agonist

α2C adrenoceptor agonist 1 is a highly selective agonist targeting the α2C-adrenoceptor, demonstrating potent activity with an EC50 value of 108 nM and a Ki of 12 nM. This compound exhibits oral bioavailability and does not penetrate the central nervous system, making it ideal for peripheral studies. Its primary application lies in the investigation of nasal congestion mechanisms and potential therapeutic interventions.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Agonist
CAS Number	928115-79-1
Applications	α2C-adrenoceptor Agonist
Formula	C₁₆H₂₁N₅O₂
Molecular Weight	315.37
SMILES	O=C(N(CC)C1=CC=C2OCCN(CC3=CN=CN3)C2=C1)NC

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.