Documents & Downloads

ABCG2-IN-5

ABCG2 Inhibitor

ABCG2-IN-5 is a selective inhibitor of the ATP-binding cassette transporter ABCG2, demonstrating an IC50 value of 0.34 µM. This compound is instrumental in investigating the mechanisms underlying ABCG2-overexpressing tumors, including non-small cell lung cancer (NSCLC). Its ability to modulate ABCG2 activity makes it a valuable tool for research focused on drug resistance and pharmacokinetics in cancer therapy.

Out of Stock

Free Aliquoting for Your Order

Tell us your preferred amount per vial. We’ll confirm the options.

Specifications

Manufacturer	Adooq Bioscience
Actions	Inhibitor
CAS Number	190323-50-3
Applications	ABCG2 Inhibitor
Formula	C₂₀H₂₂O₇
Molecular Weight	374.38
SMILES	COC1=CC(OC)=C(C(O)=C1)C(/C=C/C2=CC(OC)=C(C(OC)=C2)OC)=O

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.