Cellular Effect
| Cell Line | Activity | Value | Description | Reference |
|---|---|---|---|---|
| HEK293 | EC50 | 160 nM | Agonist activity at ferret D4 receptor in HEK293 cells coexpressing G-alpha-qo5 by FLIPR | [PMID: 17149874] |
| HEK293 | EC50 | 89 nM | Agonist activity at human D4.4 receptor in HEK293 cells coexpressing G-alpha-qo5 by FLIPR | [PMID: 17149874] |
| HEK293 | EC50 | 93 nM | Agonist activity at rat D4 receptor in HEK293 cells coexpressing G-alpha-qo5 by FLIPR | [PMID: 17149874] |