AKT inhibitor VIII (AKTI-1/2)

Catalog No.: A11286

AKT inhibitor

AKT inhibitor VIII (AKTI-1/2) Chemical Structure

CAS NO. 612847-09-3

AKT inhibitor VIII is a cell-permeable and reversible quinoxaline compound that potently and selectively inhibits Akt1/Akt2 activity (IC50 = 58 nM, 210 nM, and 2.12 μM for Akt1, Akt2, and Akt3, respectively, in in vitro kinase assays).

Availability: In stock

Package Price Qty
5 mg

Regular Price: $90.00

Special Price $72.00

10 mg

Regular Price: $140.00

Special Price $112.00

25 mg

Regular Price: $300.00

Special Price $240.00

50 mg

Regular Price: $486.00

Special Price $388.80

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

AKT inhibitor VIII is a cell-permeable and reversible quinoxaline compound that potently and selectively inhibits Akt1/Akt2 activity (IC50 = 58 nM, 210 nM, and 2.12 μM for Akt1, Akt2, and Akt3, respectively, in in vitro kinase assays).
Targets
Akt1 Akt2 Akt3
58 nM210 nM2119 nM
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 18.13 mL 90.65 mL 181.29 mL
0.5 mM 3.63 mL 18.13 mL 36.26 mL
1 mM 1.81 mL 9.06 mL 18.13 mL
5 mM 0.36 mL 1.81 mL 3.63 mL

*The above data is based on the productmolecular weight 551.6 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11286
Actions Inhibitor
M. Wt 551.6
Formula C34H29N7O
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 612847-09-3
SMILES C1CN(CCC1N2C3=CC=CC=C3NC2=O)CC4=CC=C(C=C4)C5=NC6=CC7=C(C=C6N=C5C8=CC=CC=C8)N=CN7

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