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Anticancer agent 258

Anticancer Agent

Anticancer Agent 258 is an imidazo[1,2-B][1,2,4]triazole derivative that modulates the activity of nuclear receptors. It exhibits a potent EC50 of 63 nM against Nurr in N2A cells and an impressive IC50 of 0.1 pM for Nur77 in HEK293 cells. This compound is valuable for research applications in cancer biology, metabolic disorders, and neurological diseases.

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Specifications

Manufacturer	Adooq Bioscience
CAS Number	2891984-12-4
Applications	Anticancer Agent
Formula	C₁₇H₁₂F₂N₄
Molecular Weight	310.30
SMILES	FC1=CC=C(C2=NN(C=C(N3C)C4=CC(F)=CC=C4)C3=N2)C=C1

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.