Fig. 1 · Structure
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Antitumor agent-152
Antitumor Agent
Antitumor agent-152 is a specific inhibitor of deoxycytidine kinase (dCK) that exhibits potent anticancer activity. This compound effectively hinders the uptake of tritiated deoxycytidine in L1210 leukemia cells, demonstrating an IC50 value of 1.12 μM. Antitumor agent-152 serves as a valuable tool for research applications in cancer therapies targeting nucleoside metabolism.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 1209784-87-1 |
| Applications | Antitumor Agent |
| Formula | C17H19N5O2S2 |
| Molecular Weight | 389.50 |
| SMILES | NC1=NC(SCC2=CSC(C3=CC=C(OCC)C(OC)=C3)=N2)=NC(N)=C1 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.