Fig. 1 · Structure
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APETx2
ASIC3 Inhibitor
APETx2 is a selective and reversible antagonist of the acid-sensing ion channel 3 (ASIC3), derived from the sea anemone Anthopleura elegantissima, with an IC50 of 63 nM. By targeting the external region of the ASIC3 channel, APETx2 effectively inhibits its activity. This compound demonstrates significant potential in research applications aimed at investigating mechanisms of acid-induced and inflammatory pain relief.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 713544-47-9 |
| Applications | ASIC3 Inhibitor |
| Formula | C196H280N54O61S6 |
| Molecular Weight | 4561.00 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.